SEARCH Articles Figures Tables 5-Receptor agonists pharmacological activity 5-Receptor antagonists pharmacological activity Acetylcholine receptor activation cycle Acetylcholine receptor-inducing activity Acetylcholine receptor-inducing activity ARIA) Acetylcholine receptors active site Activation of receptors Activation of the Cytoplasmic Apo-Receptor Complexes Active conformation metabotropic glutamate receptors Active receptor Active receptor Activity receptor profiling Adenosine A3 receptor activation Agonist receptor activation Agonist receptor activity Antiestrogens estrogen receptor activation mechanisms Anxiolytics serotonin receptor-active Apoptosis death receptor activation Calcitonin receptors, osteoclast activity Calcium NMDA receptor activation Calcium channels receptor-mediated activation Cannabinoid receptor constitutive activity Cell surface receptors activation Chemokine receptor activation Chemokine receptor activation, molecular Cholinergic receptors activation process Cholinergic receptors activators Cholinergic receptors structure-activity relationships Constitutive activated receptor Constitutive active receptor Constitutive active/androstane receptor Constitutive activity of receptors Constitutive androstane receptor activation Constitutive androstane receptor activators Constitutively Active Receptors and Inverse Agonists Constitutively Active Viral Chemokine Receptors Tools for Immune Subversion and Pathogenesis Constitutively activating receptor Constitutively active receptor CAR Delta receptors activation Electrochemical recognition of anionic guest species by redox-active receptor molecules Electrochemical recognition of charged and neutral guest species by redox-active receptor Electrochemical recognition of charged and neutral guest species by redox-active receptor molecules ErbB receptors activating Erythropoietin-receptor activators Estrogen receptor binding activity Estrogen receptors activity assessment Estrogen-receptors activation mechanisms Estrogen-receptors antiestrogen activity Estrogenic receptor activity Fenfluramine receptor activation Formyl peptide receptor activation Functional assays receptor activation G-protein coupled receptors activation G-protein receptors, activation G-protein-coupled receptors active GABAa receptors, activation GABAa receptors, activation barbiturate binding site GABAa receptors, activation benzodiazepine binding site GABAa receptors, activation binding affinities GABAa receptors, activation modulatory sites GABAa receptors, activation structure GABAa receptors, activation subtypes Glutamate-activated receptors H2-receptor activity Herpesviruses Encode Constitutively Active Viral Chemokine Receptors Hi-receptor activity Histamine H3 receptor, activation Histamine receptor antagonists) structure-activity relationship Hormone independent gene activation by truncated receptors Hormone-activated receptor tyrosine Hormone-activated receptor tyrosine kinase Insulin receptor activated Insulin receptor tyrosyl kinase activity Insulin receptor, activation K-Receptor agonists pharmacological activity K-Receptor antagonists pharmacological activity Kappa receptors activation Kappa-opioid receptor activation Ligand-activated nuclear receptor Ligands peroxisome proliferator-activated receptor Lumophore-spacer-receptor systems with redox active guests MSP Receptor Regulation or Activation Mechanism of Thrombin Receptor Activation Mitogen-activated protein kinase cell-surface receptors Mitogen-activated protein kinase growth factor receptor signaling Mouse vas deferens activity in receptor binding assa Mu receptors activation Muscarinic cholinergic receptors activation process Muscarinic receptors activation NMDA receptors activation NMDA receptors physiological activity Neuronal nicotinic acetylcholine receptors activation Neuronal receptors activation Nicotinic acetylcholine receptors activation mechanism Nicotinic cholinergic receptors activation process Nicotinic receptors activation Novel Receptor Active Substances Nuclear hormone receptor activator Nuclear peroxisome proliferator activated receptor Nuclear receptors, retinoid-induced gene activation Opioid receptors activation P-Opioid receptor activity in guinea-pig ileum P-Receptor agonists pharmacological activity P-Receptor antagonists pharmacological activity PEROXISOME PROLIFERATED -ACTIVATED RECEPTORS (PPARS) PPARy modulator proliferator-activated receptor PPARy, Peroxisome proliferator activated receptor gamma Partial agonism and the two-state model of receptor activation Peroxisomal proliferator-activated receptors Peroxisomal proliferator-activated receptors Subject Peroxisome Proliferator-Activated Receptor y Coactivator-la Peroxisome Proliferator-Activated Receptor y Ligands Peroxisome Proliferator-Activated Receptor y-Agonists and Stroke Peroxisome proliferation-activated receptor Peroxisome proliferation-activated receptor PPAR) Peroxisome proliferator activated receptor -a agonists Peroxisome proliferator activated receptor binding protein Peroxisome proliferator activated receptor interaction with genes Peroxisome proliferator activated receptor species difference Peroxisome proliferator activated receptor-y Peroxisome proliferator activator receptor- (PPAR Peroxisome proliferator activator receptor-a Peroxisome proliferator-activated receptor 7 agonists Peroxisome proliferator-activated receptor PPAR agonists) Peroxisome proliferator-activated receptor PPAR) Peroxisome proliferator-activated receptor PPAR) pathway Peroxisome proliferator-activated receptor PPARa activation Peroxisome proliferator-activated receptor PPARa) Peroxisome proliferator-activated receptor PPARy) Peroxisome proliferator-activated receptor PPARy) agonists Peroxisome proliferator-activated receptor action mechanisms Peroxisome proliferator-activated receptor activation Peroxisome proliferator-activated receptor agonists thiazolidinediones Peroxisome proliferator-activated receptor alpha Peroxisome proliferator-activated receptor alpha activator Peroxisome proliferator-activated receptor alpha gene Peroxisome proliferator-activated receptor alpha protein Peroxisome proliferator-activated receptor atherosclerosis Peroxisome proliferator-activated receptor balance Peroxisome proliferator-activated receptor beta Peroxisome proliferator-activated receptor chemistry Peroxisome proliferator-activated receptor effects Peroxisome proliferator-activated receptor gamma Peroxisome proliferator-activated receptor gene expression alterations Peroxisome proliferator-activated receptor human response Peroxisome proliferator-activated receptor inflammation Peroxisome proliferator-activated receptor inhibition studies Peroxisome proliferator-activated receptor insulin sensitivity improvement Peroxisome proliferator-activated receptor insulin sensitization Peroxisome proliferator-activated receptor isoforms Peroxisome proliferator-activated receptor lipid oxidation products Peroxisome proliferator-activated receptor mechanisms Peroxisome proliferator-activated receptor modulator Peroxisome proliferator-activated receptor oxidative stress Peroxisome proliferator-activated receptor pioglitazone Peroxisome proliferator-activated receptor polyunsaturated fatty acids Peroxisome proliferator-activated receptor rosiglitazone Peroxisome proliferator-activated receptor signaling Peroxisome proliferator-activated receptor target gene identification Peroxisome proliferator-activated receptor thiazolidinedione insulin sensitizers Peroxisome proliferator-activated receptor tissue expression Peroxisome proliferator-activated receptor transcriptional regulation Peroxisome proliferator-activated receptor troglitazone Peroxisome proliferator-activated receptor-alpha (PPAR Peroxisome proliferator-activated receptor-y (PPAR Peroxisome proliferator-activated receptor-y agonists Peroxisome proliferator-activated receptors Peroxisome proliferator-activated receptors PPARs), fatty acid ligands Peroxisome proliferator-activated receptors dual agonists Peroxisome proliferator-activated receptors functions Peroxisome proliferator-activated receptors structure Peroxisome proliferators activated receptor PPAR) Peroxisome proliferators activator receptor Peroxisome proliferators activator receptor PPAR) agonists Peroxisome proliferators-activated receptor Peroxisome-activator receptor-alpha Peroxisome-activator receptor-alpha expression Peroxisome-proliferator activated receptors PPARs) Platelet activating factor receptor-mediated activities Platelet activation receptors Platelet-activating factor receptor Platelet-activating factor receptor antagonists Pregnane-activated receptor Prolactin receptor activation Proliferator-activated receptor Proliferator-activated receptor PPAR)-gamma Prostanoid receptors selective ligands and structure-activity relationships Protease-activated receptor Protease-activated receptor signaling Protease-activated receptors reaction Protein tyrosine phosphorylation receptor activation Proteinase-activated receptors Quantitative structure-activity relationship estrogen receptor binding affinity Receptor Activation, Tyrosine Kinase Activity, and in Cultured Vascular Smooth Muscle Cells Receptor activation Receptor activation Receptor activation mechanism Receptor activation, molecular processes Receptor activator of NF-kB Receptor activator of NF-kB ligand Receptor activator of nuclear factor Receptor activator of nuclear factor-kB ligand Receptor activities, regulation Receptor activity dopamine Receptor activity modifying proteins Receptor activity modulating proteins Receptor activity muscarinic Receptor activity, conjugates Receptor agonists/activators Receptor binding assay activity Receptor blocking activity Receptor constitutively active Receptor destroying activity Receptor molecules, redox-active Receptor molecules, redox-active electrochemical recognition Receptor molecules, redox-active, electrochemical recognition of charged and Receptor molecules, redox-active, electrochemical recognition of charged and neutral Receptor molecules, redox-active, electrochemical recognition of charged and neutral guest Receptor molecules, redox-active, electrochemical recognition of charged and neutral guest species Receptor natural killer cells, activation Receptor signaling complexes activated Receptor tyrosine kinase Activation Receptor tyrosine kinase activity, insulin Receptor-independent activation Receptors activated solely by synthetic Receptors activated solely by synthetic ligands Receptors antitumor activity Receptors constitutive activity Receptors intrinsic enzyme activity Receptors membrane-bound, activation Receptors redox-active Receptors redox-active center Receptors with Associated Tyrosine Kinase Activity Receptors with Kinase Activity Receptors with enzymatic activity Receptors with guanylate cyclase activity Receptors with intrinsic enzymatic activity Receptors with protein kinase activity Receptors with serine/threonine kinase activity Receptors with tyrosine kinase activity Receptors without enzymatic activity Regulation of Receptor Activity Selective drugs, activity toward receptors Serotonin receptor activity Serotonin receptor-active agents Signal Transmission via Transmembrane Receptors with Tyrosine-specific Protein Kinase Activity Smad anchor for receptor activation Structural Determinants of Ligand Binding and Receptor Activation by CC Chemokines Structure-activity relationships drug-receptor interactions Structure-activity relationships of dopamine receptor agonists Structure-activity relationships receptor mapping T cell receptor activation Test Systems Addressing 5-HT4 Receptor Agonist Activity The Distinction between Agonist Binding and Receptor Activation The Estrogen Receptors and Their Multiple Gene Activation Mechanisms The Law of Mass Action, binding sites and receptors—understanding why specific, potent biological activity is a rare property for any one chemical to possess The Peroxisome Proliferator Activated Receptor The del Castillo-Katz Mechanism 1. Relationship between Agonist Concentration and Fraction of Receptors in an Active Form Thrombin receptor activation Thrombin receptor-activating peptide TRAP) Thrombin receptor-activating peptides Thromboxane receptor activation Towards electrochemical recognition of neutral guest species by redox-active receptor molecules Urokinase plasminogen activator receptor Urokinase-type plasminogen activator receptor Urokinase-type plasminogen activator receptor uPAR)