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Midazolam

The BZ stmcture also has provided a molecular scaffold for a number of peptide receptor ligands (26). Antagonists for the cholecystokinin (CCK-A) receptor, eg, devazepide (65), the thyrotropin-releasing hormone (TRH) receptor, eg, midazolam (66), and the /i -opiate receptor, eg, tifluadom (67), as well as a series of ras famyl transferase inhibitors, eg, BZA-2B (68) (30) have been identified (Table 4). [Pg.530]

Midazolam and diazepam decrease arterial pressure without a change ia heart rate. Like thiopeatoae, midazolam is a respiratory depressant. Advantages of midazolam are its amnestic effect, coupled with less postoperative depression (102). A reversal agent for the benzodiazepiaes has also become available. Flumazenil [78755-81-4] C25H24FN2O2, (5) displaces the beazodiazepiaes from their receptor but has Httie demoastrable activity of its owa (103,104). [Pg.410]

Mesoridazine besylate Methoqualone Metoclopramide HCI Metolazone Midazolam maleate Moxisylyte Nadolol Naloxone... [Pg.1609]

Mice lacking the 8 subunit, which is mainly expressed in cerebellum and thalamus, display an attenuation of ssatrighting reflex time following the administration of the neurosteroids, alphaxalone and pregnanolone, while the responses to propofol, etomindate, ketamine and the benzodiazepine midazolam were unaffected. This demonstrates the role of GABAa receptors containing the 8 subunit for neurosteroid action. [Pg.518]

Midazolam (Versed), a short-acting benzodiazepine CNS depressant, is used as a preanesthetic drug to relieve anxiety for induction of anesthesia for conscious sedation before minor procedures, such as endoscopic procedures and to supplement nitrous oxide and oxygen for short surgical procedures. When the drug is used for induction anesthesia, the patient gradually loses consciousness during a period of 1 to 2 minutes. [Pg.321]

CijHijClFNO 784-38-3) see Cinolazepam Doxefazepam Ethyl loflazepate Flunitrazepam Flurazepam Flutazolam Midazolam Quazepam... [Pg.2291]

C 5H C1FN20 2886-65-9) see Cinolazepam Doxefazepam Flutazolam Flutoprazepam Midazolam iV-[[7-chloro-5-(2-fluorophenyl)-2,3-dihydro-l r-l,4-ben-zodiazepin-2-yl]methyI]acetamide (C,sH,7C1FN20 59467-68-4) see Midazolam... [Pg.2329]

CH3NO2 75-52-5) see Baclofen Gabapentin Midazolam Pirbuterol Ranitidine Ropinirole Trometaniol l-(2-nitro-4-methoxyphenyl)-2-nitropropcnc C oHi()N203 25803-11-6) see Clometacin 4-(5-nitro-l-methylindol-3-ylmethyl)-3-methoxybenzoic acid... [Pg.2426]

Ator NA Relation between discriminative and reinforcing effects of midazolam, pentobarbital, chlordiazepoxide, Zolpidem, and imidazenil in baboons. Psychopharmacology (Berl) 163 477 87, 2002... [Pg.148]


See other pages where Midazolam is mentioned: [Pg.635]    [Pg.635]    [Pg.635]    [Pg.528]    [Pg.410]    [Pg.223]    [Pg.223]    [Pg.223]    [Pg.223]    [Pg.227]    [Pg.257]    [Pg.272]    [Pg.1024]    [Pg.1613]    [Pg.1694]    [Pg.1694]    [Pg.1707]    [Pg.1743]    [Pg.129]    [Pg.133]    [Pg.139]    [Pg.253]    [Pg.563]    [Pg.1137]    [Pg.319]    [Pg.321]    [Pg.324]    [Pg.407]    [Pg.1328]    [Pg.1328]    [Pg.2280]    [Pg.2329]    [Pg.2329]    [Pg.2329]    [Pg.2329]    [Pg.2380]    [Pg.2411]    [Pg.120]    [Pg.125]    [Pg.126]   
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Ciclosporin Midazolam

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Diclofenac Midazolam

Echinacea Midazolam

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Fentanyl midazolam

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Foods: Grapefruit juice Midazolam

Halothane midazolam

Hormonal) Midazolam

Hydroxy midazolam

Hypotension midazolam

Imatinib Midazolam

Isoflurane midazolam

Ketoconazole midazolam

Lidocaine Midazolam

Look up the names of both individual drugs and their drug groups to access full information Midazolam

Medicines) Midazolam

Mepivacaine Midazolam

Metabolism midazolam

Methadone Midazolam

Methylphenidate Midazolam

Methylprednisolone Midazolam

Midazolam Alcohol

Midazolam Aminophylline

Midazolam Aspirin

Midazolam Atracurium

Midazolam Bupivacaine

Midazolam CYP3A4/5/7 substrate

Midazolam Calcium-channel blockers

Midazolam Carbamazepine

Midazolam Clarithromycin

Midazolam Corticosteroids

Midazolam Cyclosporine

Midazolam Erythromycin

Midazolam Ethanol

Midazolam Fluconazole

Midazolam Fluoxetine

Midazolam Fosphenytoin

Midazolam Itraconazole

Midazolam Metronidazole

Midazolam Morphine

Midazolam Nitrendipine

Midazolam Pancuronium

Midazolam Phenytoin

Midazolam Prednisolone

Midazolam Propofol

Midazolam Ranitidine

Midazolam Rifampin

Midazolam Rimonabant

Midazolam Sevoflurane

Midazolam Succinylcholine

Midazolam Sufentanil

Midazolam Suxamethonium

Midazolam Tacrolimus

Midazolam Tadalafil

Midazolam Terbinafine

Midazolam Tetracaine

Midazolam Theophylline

Midazolam Thiopental

Midazolam Tobacco

Midazolam Valerian

Midazolam Valproate

Midazolam Vecuronium

Midazolam Verapamil

Midazolam acidosis

Midazolam adverse effects

Midazolam agitation

Midazolam anesthesia

Midazolam antifungal azoles

Midazolam apnea with

Midazolam atorvastatin

Midazolam azithromycin/clarithromycin

Midazolam cardiovascular

Midazolam clearance

Midazolam comparative studies

Midazolam critical care

Midazolam desaturation

Midazolam diltiazem

Midazolam dizziness

Midazolam dosage

Midazolam dosing

Midazolam drug administration

Midazolam drug administration route

Midazolam drug interactions

Midazolam drug overdose

Midazolam effect

Midazolam for

Midazolam grapefruit juice

Midazolam hiccups

Midazolam hydrochloride

Midazolam hydroxylation activity

Midazolam induction

Midazolam interactions

Midazolam intranasal administration

Midazolam macrolides

Midazolam maleate

Midazolam nervous system

Midazolam nitrous oxide

Midazolam observational studies

Midazolam pethidine

Midazolam pharmacokinetics

Midazolam placebo-controlled studies

Midazolam poisoning with

Midazolam protease inhibitors

Midazolam quantitation

Midazolam reduction

Midazolam respiratory

Midazolam rifampicin

Midazolam saquinavir

Midazolam status epilepticus

Midazolam systemic clearance

Midazolam toxicity

Midazolam with itraconazole

Midazolam with protease inhibitors

Midazolam with telithromycin

Nefazodone midazolam

Paediatrics midazolam

Sedation-induction midazolam

Sedative Hypnotics midazolam

T- Midazolam

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