Gamma aminobutyric acid receptor

Miller LG, Greenblatt DJ, Roy RB, et al Chronic benzodiazepine administration, II discontinuation syndrome is associated with upregulation of gamma-aminobutyric acid receptor complex binding and function. J Pharmacol Exp Ther 246 177-182, 1988b... [Pg.157]

Corrigall WA et al. Response of nicotine self-administration in the rat to manipulations of mu-opioid and gamma-aminobutyric acid receptors in the ventral tegmental area. Psychopharmacology 2000 149(2) 107-114. [Pg.459]

Abalis IM, Eldefrawi AT, Eldefrawi ME (1986) Actions of avermectin Bla on the gamma-aminobutyric acid receptor and chloride channels in rat brain. J Biochem Toxicol 1 69-82... [Pg.72]

DE GAMMA-AMINOBUTYRIC-ACID RECEPTOR PI SUBUNIT PRECURSOR (GABA(A)... [Pg.62]

GABRP Gamma-aminobutyric acid receptor pi subunit... [Pg.259]

Cui Y, Rajasethupathy P, Hess GP (2004) Selecrion of stable RNA molecules that can regulate the channel-opening equilibrium of the membrane-bound gamma-aminobutyric acid receptor. Biochemistry 43 16442-16449... [Pg.38]

Mectianism of Action An antidote that antagonizes the effect of benzodiazepines on the gamma-aminobutyric acid receptor complex in the CNS. Therapeutic Effect Reverses sedative effect of benzodiazepines. [Pg.507]

Susdak PD, Schwartz RD, Scolnick P, et al Ethanol stimulates gamma-aminobutyric acid receptor-mediated chloride transport in rat brain synaptoneurosomes. Proc Natl Acad Sci U S A 83 4071-4075, 1986... [Pg.753]

W Chen, M Terada, JT Cheng. Characterization of subtypes of gamma-aminobutyric acid receptors in an Ascaris muscle preparation by binding assay and binding of PF1022A, a new anthelmintic, on the receptors. Parasitol Res 82 97-101, 1996. [Pg.495]

Kuriyama, T., Schmidt, T.J., Okuyama, E. and Ozoe, Y. (2002) Structure-activity relationships of seco-prezizaane terpenoids in gamma-aminobutyric acid receptors of houseflies and rats. Bioorganic and Medicinal Chemistry 1 0(6), 1 873-1 881. [Pg.329]

Zheng W, Xie W, Zhang J, Strong JA, Wang L, Yu L, Xu M, Lu L (2003) Function of gamma-aminobutyric acid receptor/channel rho 1 subunits in spinal cord. J Biol Chem 278 48321-48329... [Pg.535]

Twyman, R.E., Rogers, C.J., and MacDonald, R.L., 1989. Differential regulation of gamma aminobutyric acid receptor channels by diazepam and phenobarbital, Ann. Neurol, 25, pp. 213-220. [Pg.157]

Fritschy JM, Benke D, Mertens S, Oertel WH, Bachi T, et al. 1992. Five subtypes of type A gamma-aminobutyric acid receptors identified in neurons by double and triple immunofluorescence staining with subunit-specific antibodies. Proc Natl Acad Sci USA 89 6726-6730. [Pg.188]

Maestrini E, Lai C, Marlow A, Matthews N, Wallace S, Bailey A, Cook EH, Weeks DE, Monaco AP (1999) Serotonin transporter (5-HTT) and gamma-aminobutyric acid receptor subunit beta3 (GABRB3) gene polymorphisms are not associated with autism in the IMGSA families. The International Molecular Genetic Study of Autism Consortium. Am J Med Genet 88 492 96. [Pg.124]

Martin ER, Menold MM, Wolpert CM, Bass MP, Donnelly SL, Ravan SA, Zimmerman A, Gilbert JR, Vance JM, Maddox LO, Wright HH, Abramson RK, DeLong GR, Cuccaro ML, Pericak-Vance MA (2000) Analysis of linkage disequilibrium in gamma-aminobutyric acid receptor subunit genes in autistic disorder. Am J Med Genet 96 43-48. [Pg.124]

Abbreviations AOB, accessory olfactory bulb mAChR, muscarinic cholinergic receptor nAChR, nicotinic cholinergic receptor alpha and beta adrenergic receptors D, dopamine receptors 5-HT,a and S-HTja/c, serotonin receptors NMDA, N-methyl-D-Aspartate receptor AMPA, a-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor GABAa/b, gamma aminobutyric acid receptor XX, receptor present in region. [Pg.538]

Zaleplon is a sedative and hypnotic that interacts with the gamma-aminobutyric acid-receptor complex. It is indicated in the short-term treatment of insomnia. [Pg.741]

Lawrence LJ, Casida JE (1983) Stereospecific action of pyrethroid insecticides on the gamma-aminobutyric acid receptor-ionophore complex. Science 221 1399... [Pg.3284]

Crofton KM, Reiter LW (1987) Pyrethroid insecticides and the gamma-aminobutyric acid receptor complex Motor activity and the acoustic startle response in the rat. J Pharmacol Exp... [Pg.3284]

A team at Merck, in 2005, used the Suzuki-Miyaura reaction as a key step in the synthesis of an orally active 2/3-selective GABAA (Gamma-aminobutyric acid receptor) agonist candidate for the treatment of centrtJ nervous system conditions (Scheme 1.43) [143]. The biaryl product was crystallized from water/t-PrOH in 85% and it had a purity of 96.3% (HPLC). [Pg.64]

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