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Receptors androgen

Androgens, namely testosterone and dihydrotestosterone (DHT), are involved in growth and maintenance of the prostate gland. Testosterone and DHT exert their effect [Pg.779]

The first crystal structure of the LED of the AR in complex with metri-bolone (R1881) was solved by Matias and colleagues in 2000 [38]. The LED has a similar three-dimensional structure to the other agonist-bound steroid receptors, namely the ERa, ERj6 and the PR [38]. The fact that all steroid hormone receptors bind similar hormone response elements (HREs) stands in sharp contrast to the specific activities elicited by application of the steroid [Pg.28]


Androgen receptor binding/Reporter gene assay. [Pg.18]

The mechanism by which TBT causes these effects has been extensively stiidied. The androgenic effects of TBT appear to be caused by interference with steroid biosynthesis rather than by mimicking the action of testosterone at the androgen receptor. Exposure of female molluscs to TBT leads to an elevation in testosterone in the haemolymph. " Much of the experimental evidence... [Pg.56]

Sex Steroid Receptors Androgen Receptor, Estrogen Receptors, Progesterone Receptor... [Pg.75]

Hormone antagonists (tamoxifen and toremifen bind to the estradiol receptor, flutamide binds to the androgen receptor) are used for treating breast and prostate cancer. [Pg.155]

Androgen receptor Transcriptional regulator Inhibition of androgen receptor transcriptional activity... [Pg.187]

Sex steroid receptors are members of the steroid hormone receptor (SHR) family that ligand-dependently regulate functions of the sexual organs. Sex steroid receptors are the androgen receptor [1] (AR), the estrogen receptor a [2] and (3 [3] (ERa, ER 3), and the progesterone receptor [4] (PR). [Pg.1126]

Sex Steroid Receptors Androgen Receptor, Estrogen Receptors, Progesterone Receptor. Figure 1 Schematic structures of AR, ERa, ER(3, and PR. [Pg.1127]

OMIM (Online Medelian Inheritance in Man) www. ncbi.nlm.nih.gov/entrez 313700 ANDROGEN RECEPTOR AR... [Pg.1130]


See other pages where Receptors androgen is mentioned: [Pg.220]    [Pg.222]    [Pg.89]    [Pg.93]    [Pg.97]    [Pg.102]    [Pg.107]    [Pg.65]    [Pg.80]    [Pg.80]    [Pg.894]    [Pg.977]    [Pg.1063]    [Pg.1078]    [Pg.1092]    [Pg.1110]    [Pg.1112]    [Pg.1113]    [Pg.1117]    [Pg.1117]    [Pg.1127]   
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AR, Androgen receptor

Androgen Receptor Complexes

Androgen receptor aberrations

Androgen receptor affinity

Androgen receptor antagonists

Androgen receptor antagonists steroidal

Androgen receptor binding

Androgen receptor blockers

Androgen receptor gene amplification

Androgen receptor modulators

Androgen receptor mutations

Androgen receptor phosphorylation

Androgen receptor prostate cancer

Androgen receptor protein

Androgen receptor structure

Androgen receptor therapeutic modulation

Androgen receptor, in prostate cancer

Androgen receptor, pesticide binding

Androgenic receptor

Androgenization

Androgens

Androgens brain receptors

Cancer androgen receptor

Markers androgen receptor

Nonsteroidal Tissue-selective Androgen Receptor Modulators

Nonsteroidal androgen receptor agonists

Nonsteroidal androgen-receptor antagonists

Nuclear androgen receptors

Receptor androgen, binding affinity

Receptors SARM (selective androgen

Receptors androgen receptor

Selective Androgen Receptor Modulator

Selective androgen receptor

Selective androgen receptor modulators

Selective androgen receptor modulators SARMs)

Sex Steroid Receptors: Androgen Receptor, Estrogen

Spironolactone androgen receptors inhibited

Steroid androgen receptor

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