Thyrotropin-releasing hormone analogs

Colson AO, Gershengorn MC. Thyrotropin-releasing hormone analogs. Mini Rev Med Chem. 2006 6 221-226. 

C., and Moeller, K. D. (1998) Thyrotropin releasing hormone analogs A building block approach to the construction of tetracyclic peptidomimetics. Bioorg. Med. Chem. Lett. 8, 3093-3096. 

Nemeroff CB, Bissette G, Martin JB, et al Effect of chronic treatment with thyrotropin-releasing hormone (TRH) or an analog of TRH (hnear-beta-alanine TRH) on the hypothalamic-pituitary-thyroid axis. Neuroendocrinology 30 193-199, 1980... 

Simulated annealing has also been applied to the conformational study of dipeptide models of Gly, Ala, and Asp pentaglycine and Leu-enkephalin [11] an analog of vasopressin [10] (3S, 4S)-statin [12] analogs of thyrotropin releasing hormone [13] and the C-peptide of Ribonuclease A [13]. 

TRH Analogs. A similar strategy was used 56-359) for the CNS delivery of a thyrotropin-releasing hormone (TRH, Glp-His-Pro) analog (Glp-Leu-Pro) in which histidine (His ) was replaced with leucine (Leu )to... 

Monga V, Meena CL, Kaura N, Jain R (2008) Chemistry and biology of thyrotropin-releasing hormone (TRH) and its analogs. Curr Med Chem 15 2718—2733... 

Drug Design and the Receptor-Bound Conformation of Thyrotropin Releasing Hormone (TRH) Design and Synthetic Approaches Towards Rigid TRH Analogs. 

Yokohama, S., Yoshioka, T., and Kitamoii, N., 1984a, Absorption ofg-butyrolactone-g-carbon-yl-L-histidyl-L-prolinamide citrate (DN-1417), an analog of thyrotropin-releasing hormone, in rats and dogs. J. Pharmacobio-Dyn. 7 527-535. 

Hichens M. A comparison of thyrotropin-releasing hormone with analogs Influence of disposition upon pharmacology. Drug Metab Rev. 1983 14(l) 77-98. 

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