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Imidazoline receptor ligands

Holt A, Wieland B, Baker GB. 2004. Allosteric modulation of semicarbazide-sensitive amine oxidase activities in vitro by imidazoline receptor ligands. Br J Pharmacol 143 495. [Pg.132]

Discovery of Highly Selective Imidazoline Receptor Ligands... [Pg.361]

Brasili L, Pigini M, Bousquet P, Carotti A, Dontenwill M, Giannella M, Moriconi R, Piergentili A, Quaglia W, Tayebati SK Discovery of highly selective imidazoline receptor ligands... [Pg.422]

Milligan, C.M., MacKinnon, A.C., 1997. Imidazoline receptor ligands. Drugs New Perspect. 10, 74-84. [Pg.134]

Discovery of highly selective imidazoline receptor ligands. Perspective in Receptor Research 24, 361-376. [Pg.139]

In medicinal applications, l,2,3,4-tetrahydropyrazino[l,2-alindoles were of interest as high-affinity selective imidazoline receptor ligands <04BMCL1003>, 3,4-dihydro-l//-pyrido[2,3-l ]-pyrazin-2-ones as corticotropin-releasing factor-1 (CRF 1) receptor antagonists <04JMC5783>,... [Pg.327]

Chan, S.L., Atlas, D., James, R.F. and Morgan, N.G. (1997) The effect of the putative endogenous imidazoline receptor ligand, clonidine-displacing substance, on insulin secretion from rat and human islets of Langerhans. Br. J. Pharmacol. 120 926-932. [Pg.300]

Pharmacophore development and SAR studies of imidazoline receptor ligands 12MRM1542. [Pg.283]

Prisinzano T, Dukat M, Law H, et al. 2-(Anilino)imidazolines and 2-(benzyl)-imidazoline derivatives as /z5-HT1D serotonin receptor ligands. Bioorg Med Chem Lett 2004 14 4697-4699. [Pg.141]

In some instances, very slight changes such as hydrogenation or dehydrogenation can indnce dramatic changes in the activity profile of drug molecules. Examples are found in the imidazoline I3 receptor ligands which act on... [Pg.422]

Chart 1. Some of the most used ligands for imidazoline receptors characterization. [Pg.362]

Regunathan, S., Reis, D.J., 1996. Imidazoline receptors and their endogenous ligands. Ann. Rev. Pharmacol. Toxicol. 36. 511-544. [Pg.134]

LNP 509), an 1] imidazoline receptor selective ligand with hypotensive activity. Journal of Medicinal Chemistry, 44, 1588-1593. [Pg.28]

Karolak-Wojdechowska, J., Kiec-Kononowicz, K., and Mrozek, A. (2001) Structure and activity studies of glycine receptor ligands. Part 7. Structural remarks on arylidene-imidazoline-4-one glycinates and glydnamides. Journal of Molecular Structure, 597, 73-81. [Pg.100]

Imidazolines have been shown to have biological utility as antidepressants, and imidazoline ligands are known for a number of receptors widely distributed in both the peripheral and central nervous system.39 The imidazoline moiety has also been extensively studied as an amide bond... [Pg.480]

One of the latest theories to account for the action of bupropion is its influence on imidazoline I, receptors. Agmatine (decarbosylated arginine) may be an endogenous ligand for I, sites. Evidence indicates that plasma agma-... [Pg.515]

See other pages where Imidazoline receptor ligands is mentioned: [Pg.489]    [Pg.52]    [Pg.173]    [Pg.171]    [Pg.570]    [Pg.52]    [Pg.563]    [Pg.353]    [Pg.355]    [Pg.364]    [Pg.2]    [Pg.134]    [Pg.134]    [Pg.295]    [Pg.563]    [Pg.177]    [Pg.11]    [Pg.45]    [Pg.45]    [Pg.259]    [Pg.355]    [Pg.357]    [Pg.361]    [Pg.372]    [Pg.100]    [Pg.108]    [Pg.132]    [Pg.285]    [Pg.1151]   
See also in sourсe #XX -- [ Pg.361 , Pg.362 , Pg.363 , Pg.364 , Pg.365 , Pg.366 , Pg.367 , Pg.368 , Pg.369 , Pg.370 , Pg.371 ]



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Imidazoline

Imidazoline receptors

Receptor ligands

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