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Opioid receptors ligands

In an approach to opioid receptor ligands,diazabicyclononanones were prepared in a double Petrenko-Kritschenko reaction. Diester 76, in the presence of methylamine and aryl aldehydes, was converted to piperidone 77. This was immediately resubmitted to the reaction conditions however, in this iteration formaldehyde replaced the aryl aldehyde component. The outcome of this reaction produced 78 which was further investigated for its use in rheumatoid arthritis. [Pg.313]

Molecular modelling of opioid receptor-ligand complexes, 40 (2002) 107 Molecularly imprinted polymers,... [Pg.389]

Meng F, Ueda Y, FIoversten MT et al. Mapping the receptor domains critical for the binding selectivity of d-opioid receptor ligands. Eur J Pharmacol 1996 311 285-292. [Pg.487]

Two artificial compound libraries were chosen as compound mixtures, of which library 1 was composed only of dummy ligands (acetanilide, amitryptiline, benzoic acid, (+)-bicuculline, 4-chloraniline, 2,3-dichloraniline, methylbenzoate, phenol, tramadol see Fig. 7.11), whereas library 2 contained, in addition to these compounds, naloxone, a known //-opioid receptor ligand. [Pg.264]

Shippenberg TS, Herz A Influence of chronic lithium treatment upon the motivational effects of opioids alteration in the effects of mu- but not kappa-opioid receptor ligands. J Pharmacol Exp Ther 256 1101-1106, 1991 Shippenberg TS, Millan MJ, Mucha RE, et al Involvement of beta-endorphin and mu-opioid receptors in mediating the aversive effect of lithium in the rat. Eur J Pharmacol 154 135-144, 1988... [Pg.744]

Dooley, C., Houghten, R. (1993) The use of positional scanning synthetic peptide combinatorial libraries for the rapid determination of opioid receptor ligands. Life Sci 52, 1509-1517. [Pg.24]

Dooley, C. and Houghten, R. (Torrey Pines Institute for Molecular Studies) Novel mu opioid receptor ligands agonists and antagonists, W09640208 (1996) US5641861 (1997) US5919897 (1999). [Pg.157]

Grandy, D.K., Bunzow, J.R., Civelli, O., Reinscheid, R.K., Nothacker, H.-P., Monsma, F.J. (Oregon Health Sciences University) Mammalian opioid receptor ligand and uses, US5837809 (1975). [Pg.157]

Putz, C.K., Straliburger, W., Zimmer, O., Englberger, W. (Grunenthal GmbH) Preparation of aryltetrahydroacridinemethanamines as S-opioid receptor ligands, EP970949 (1998). [Pg.466]

TABLE 1 Binding Affinities for Selective Opioid Receptor Ligands to Membrane Preparations from COS-7 Cells, Transiently Transfected with the Cloned Human Delta Opioid Receptor... [Pg.36]

Benzhydrylpiperazines as Nonpeptidic Delta Opioid Receptor Ligands... [Pg.113]

The structural class of piperazinyl benzamides contains a number of SNC80-like delta opioid receptor ligands. These compounds have been... [Pg.366]

INTRACELLULAR SIGNALING MECHANISMS UPON OPIOID RECEPTOR LIGAND BINDING... [Pg.386]

Teschemacher, H., Koch, G., and Brantl, V. 1997. Milk protein-derived opioid receptor ligands. Biopolymers 43, 99—117. [Pg.273]

Synthesis of fluorine-18 labelled kappa opioid receptor ligands... [Pg.422]

See other pages where Opioid receptors ligands is mentioned: [Pg.259]    [Pg.76]    [Pg.32]    [Pg.156]    [Pg.92]    [Pg.711]    [Pg.457]    [Pg.457]    [Pg.465]    [Pg.116]    [Pg.25]    [Pg.25]    [Pg.114]    [Pg.115]    [Pg.115]    [Pg.163]    [Pg.163]    [Pg.332]    [Pg.342]    [Pg.432]    [Pg.433]    [Pg.435]    [Pg.435]    [Pg.435]    [Pg.468]    [Pg.48]    [Pg.231]    [Pg.186]    [Pg.259]    [Pg.259]    [Pg.260]    [Pg.262]    [Pg.264]    [Pg.266]   
See also in sourсe #XX -- [ Pg.315 ]

See also in sourсe #XX -- [ Pg.259 , Pg.262 , Pg.265 , Pg.273 ]

See also in sourсe #XX -- [ Pg.5 , Pg.374 , Pg.375 ]

See also in sourсe #XX -- [ Pg.5 , Pg.374 , Pg.375 ]



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Delta opioid receptor ligands

Endogenous opioid receptor ligand

Opioid receptors

Opioid receptors ligand binding model

Opioids receptors

Receptor ligands

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