2- indoles, synthesis from

Aniline, N-alkyl-o-allyl-indole synthesis from, 4, 321 Aniline, N-allyl-... 

Ethoheptazine as analgesic, 1, 167 Ethosuximide as anticonvulsant, 1, 166 Ethoxzolamide as diuretic, 1, 173 Ethylamine, o-bromophenyl-indole synthesis from, 4, 322 Ethylamine, 2-thienyl-biological activity, 4, 911 Ethylamine, 3-thienyl-biological activity, 4, 912 Ethylene... 

New Indole Chemistry from Development of Pd Chemistry 4.2.2.1 Discovery of New Indole Synthesis from Amines... 

For a general, simple high yield indole synthesis from anilines and methylthioacetaldehyde etc. see JACS 95,588,591,2718,6508 (1973). For indoles from N-( /3 -hydroxy-ethyl aniline esters see BSC 2485(1973). For a 2-acyl-indoles in one step from orthoamino-ketones and alpha-haloketones or 2-carboxyindoles from sulfonamides of ortho-aminocarbonyls see JOC 38,3622-24(1972). Indole and 5-Br-indole in 4 steps from beta-naphthol see Chem. Het. Cpds. (Russ.) 753(1973). Indole-JOC 37,3622(1972). 

Among early reported Pd-catalyzed reactions, the Mori-Ban indole synthesis has proven to be very useful for pyrrole annulation. In 1977, based on their success of nickel-catalyzed indole synthesis from 2-chloro-fV-allylaniline, the group led by Mori and Ban disclosed Pd-catalyzed intramolecular reactions of aryl halides with pendant olefins [122]. Compound 102, easily prepared from 2-bromo-lV-acetylaniline and methyl bromocrotonate, was adopted as the cyclization precursor. Treatment of 102 with Pd(OAc)2 (2 mol%), Ph3P (4 mol%) and NaHCQ3... 

Ilac Fischer indole synthesis from /V-arylhydrazones 3.06.3.4.2... 

Processes include the Fischer indole synthesis from arylhydrazones and related sigmatropic syntheses, reductive evclizations of nitni compounds, the Madelung synthesis from anilides and related base-cululyxed condensations. and transition-metal catalyzed cyclizations,... 

Benzophenone, o-benzoylamino-indole synthesis from, 4, 329 Benzophenone, 2,3 -dihydroxy-cyclization, 3, 835... 

NENITZESCU Indole Synthesis Indole synthesis from quinones and anwio crotonates... 

BISCHLER - MOHLAU Indole synthesis Indole synthesis from a aminoacetophenones... 

Aniline, JV-alkyl-o-allyl-indole synthesis from, 4, 321 Aniline, N-allyl-indole synthesis from, 4, 326 Aniline, AT-allyl-o-bromo-indole synthesis from, 4, 327 Aniline, N-allyl-o-iodo-indole synthesis from, 4, 327 Aniline, o-bromo-in indole synthesis, 4, 340 Aniline, o-halo-cyclization, 4, 340 Aniline, m-nitro-in indole synthesis, 4, 338 Aniline black, 3, 197 Anilines... 

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