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Drug bioavailability

Because of its convenience and good patient compliance, oral administration is the most preferred drug delivery form. As a result, much of the attention of in silico approaches is focused on modeling drug oral absorption, which mainly occurs in the human intestine. In general, drug bioavailability and... [Pg.498]

Agoram B, Woltosz WS and Bolger MB. Predicting the impact of physiological and biochemical processes on oral drug bioavailability. Adv Drug Deliv Rev 2001 50 Suppl l S41-67. [Pg.509]

Chan, O. H., Stewart, B. H. Physicochemical and drug-delivery considerations for oral drug bioavailability. Drug Discov. Today 1996, 1, 461 73. [Pg.46]

Avdeef, A. High-throughput Measurement of Membrane Permeability. In Drug Bioavailability (Methods and Principles in Medicinal Chemistry), Van de Waterbeemd, H Lennemas, H Armrsson, P. (eds.), Wiley-VCH, Weinheim, 2003, pp. 46-71. [Pg.80]

A good deal of attention recently has been directed towards the use of derivatives of cyclodextrin for the solubilization and stabilization of pharmaceuticals [124 126]. One cautionary note—complexation may adversely affect the dissolution an/or permeability characteristics of the drug, thereby possibly decreasing drug bioavailability. [Pg.166]

Figure 7.15 Kinetics of transport across a filter-immobilized artificial membrane (a) desipramine and (b) dihydromethysticin concentrations in acceptor well. [Reprinted from Avdeef, A., in van de Waterbeemd, H. Lennemas, H. Artursson, R (Eds.). Drug Bioavailability. Estimation of Solubility, Permeability, Absorption and Bioavailability. Wiley-VCH Weinheim, 2003 (in press), with permission from Wiley-VCH Verlag GmbH.]... Figure 7.15 Kinetics of transport across a filter-immobilized artificial membrane (a) desipramine and (b) dihydromethysticin concentrations in acceptor well. [Reprinted from Avdeef, A., in van de Waterbeemd, H. Lennemas, H. Artursson, R (Eds.). Drug Bioavailability. Estimation of Solubility, Permeability, Absorption and Bioavailability. Wiley-VCH Weinheim, 2003 (in press), with permission from Wiley-VCH Verlag GmbH.]...
VHL Lee, KW Morimoto, RE Stratford Jr. (1982). Esterase distribution in the rabbit cornea and its implications in ocular drug bioavailability. Biopharm Drug Dispos 3 291-300. [Pg.377]

Drug Bioavailability Estimation of Solubility, Permeability, Absorption and Bioavailability. Edited by Han van de Waterbeemd. Hans Lennernas and Per Artursson Copyright 2003 WILEY-VCH Verlag GmbH Co. KGaA, Weinheim ISBN 3-527-30438-X... [Pg.2]

The Importance of Cut Wall Metabolism in Determining Drug Bioavailability... [Pg.311]


See other pages where Drug bioavailability is mentioned: [Pg.235]    [Pg.432]    [Pg.64]    [Pg.194]    [Pg.241]    [Pg.422]    [Pg.459]    [Pg.462]    [Pg.465]    [Pg.207]    [Pg.333]    [Pg.361]    [Pg.363]    [Pg.116]    [Pg.267]   
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See also in sourсe #XX -- [ Pg.4 , Pg.16 , Pg.390 , Pg.393 ]




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Bioavailability drug absorption

Bioavailability drug administration routes

Bioavailability drug delivery

Bioavailability drug discovery process

Bioavailability drug dissolution

Bioavailability drug formulations

Bioavailability drug-likeness

Bioavailability enhancement drug delivery systems

Bioavailability generic drug product

Bioavailability generic drugs

Bioavailability of a drug

Bioavailability of drugs

Bioavailability plasma drug concentrations

Bioavailability studies immediate-release drug product

Bioavailability testing drug product selection

Bioavailability, enhanced drug-dosage forms

Bioavailability, oral drugs

Complex drug substances, bioavailability

Computational Approaches to Drug Absorption and Bioavailability

Drug administration bioavailability

Drug bioavailability digoxin

Drug bioavailability improvement, methods

Drug bioavailability improvement, methods system

Drug compounds oral bioavailability

Drug development oral bioavailability

Drug discovery bioavailability

Drug product bioavailability

Drug substance bioavailability

Emulsion drug bioavailability

Generic drug products bioavailability-bioequivalency

Hydrophobic drugs bioavailability

Lipophilic drugs bioavailability

Local drug bioavailability

Long-half-life drugs, bioavailability

Oral administration bioavailability, drug-likeness

Oral drug absorption bioavailability

Oral drug delivery bioavailable dose

Orally administered drugs bioavailability

Plasma drug concentrations relative bioavailability

Profiling the Effect of Food on Drug Bioavailability

Pulmonary drug delivery oral bioavailability

Soluble drugs, poorly bioavailability

The Importance of Gut Wall Metabolism in Determining Drug Bioavailability

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