Cyclooxygenase 1/2 inhibitors NSAIDs

Benoral benorylate. benorilate benorylate. benorylate [ban] (benorilate [inn] paracetamol acetylsallcylate BenoraP ) is an aspirin-paracetamol ester, and these two pharmacologically active constituents are released systemically at different rates. It has cyclooxygenase inhibitor, nsaid analgesic, antiinflammatory and antirheumatic activity. It is used orally, particularly to treat the pain of rheumatic disease and other musculoskeletal disorders, as well as to treat fever, benoxaprofen [ban, inn, usan] (Opren ) is one of the propionic acid series of CYCLOOXYGENASE INHIBITORS with nsaid ANALGESIC. ANTIINFLAMMATORY and ANTIPYRETIC activity also effective for psoriasis. It was withdrawn due to adverse drug reactions. 

Several interesting findings dealing with 2-quinolinylmethyl esters related to Rev 5901A (139) have been reported. Workers at Wyeth-Ayerst found that attachment of this moeity to a number of classical NSAIDs endowed these cyclooxygenase inhibitors with 5-LO inhibitory activity in cell assays... 

W 7320) is one of the heteroaryl acetic acid series of CYCLOOXYGENASE INHIBITORS with NSAID ANALGESIC,... 

Amidone methadone, amidopyrine (aminophenazone [inn] and many other names) is one of the pyrazone series of CYCLOOXYGENASE INHIBITORS with NSAID ANALGESIC. ANTIINFLAMMATORY and ANTIPYRETIC activity. The risk of agranulocytosis is high and so it is rarely used. It has been used as the cyclamate salt, aminophenazone cyclamate [inn], and the butyl iodide, butopyrammonium iodide [inn]. amifenazole amiphenazole. amifloxacin [ban, inn. usan] (amifloxacln mesylate [usan]) is a fluoroquinolone derivative with antibacterial properties. 

Clonitazene [ban. inn) (Ciba 19390 NIH 7586) is a benzimidazole derivative, an opioid receptor antagonist. Clonixin [inn, usan) (CBA 93626 Sch 10304) is a pyridinecarboxylic acid derivative, a CYCLOOXYGENASE INHIBITOR With NSAID ANALGESIC. ANTIINFLAMMATORY and ANTIPYRETIC activity. It is also used in the form of a lysine salt, lysine clonixinate also the dihydroxypropyl ester, clonixeril [inn, usan). 

It can be used orally to treat infection by the herpes viruses, famotidine [ban. inn, usan[ (YM 11170 L 643341 MK 208 Pepcid ) is a thiosulfamoylpropionamidine, a histamine Hj-RECEPTOR ANTAGONIST. It is a GASTRIC SECRETION INHIBITOR and ANTIULCEROGENIC. It is also suggested to be beneficial in the treatment of schizophrenia, and as an antiviral. famprofazone [ban. inn] is one of the pyrazolone series of cyclooxygenase inhibitors with nsaid analgesic. 

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