4-Aminocarbonyl-3- 2-hydroxy-2- -ethyl

For a general, simple high yield indole synthesis from anilines and methylthioacetaldehyde etc. see JACS 95,588,591,2718,6508 (1973). For indoles from N-( /3 -hydroxy-ethyl aniline esters see BSC 2485(1973). For a 2-acyl-indoles in one step from orthoamino-ketones and alpha-haloketones or 2-carboxyindoles from sulfonamides of ortho-aminocarbonyls see JOC 38,3622-24(1972). Indole and 5-Br-indole in 4 steps from beta-naphthol see Chem. Het. Cpds. (Russ.) 753(1973). Indole-JOC 37,3622(1972). 

Sulfimid N-Aminocarbonyl-S,S-dimethyl- Ell, 905 [(H3C)2S + Hamstoff) IsothioharnstofT S-(2-Hydroxy-ethyl)- (Hydrochlorid) IX, 902... 

Imidazol 4-Aminocarbonyl-5-[3-(2-hydroxy-ethyl)-3-methyl-l -triazeno]- E16a, 1200 (Het — N + Amin)... 

Hydrazin l,2-Bis- [2-ch or-l-(chlor-difluor-methyl)-2,2-difluor-l-hydroxy-ethyl]-aminocarbonyl -E14a/2, 63 (Keton/Harnstoff)... 

S,4S)-4-Benzoyl-3-[(/ )-l-hydroxy-ethyl]-2-oxo- E16b, 189 (aus Aminocarbonyl-oxiran)... 

Bleomycin Bleomycin is a stereoisomer of 6-amino-A-[[2-[[4-[[l-[[[2-[4-(aminocar-bonyl)[2,4i-bintiazol]-2i-yl]ethyl]amino]carbonyl]-2-hydroxypropylamino-2-hydroxy-l,3-dimethyl-4-oxobutyl]amino-l-[[2-0-[3-0-(aminocarbonyl)-a-D-... 

Aminocarbonyl-ethyl)-dibenzyl- XII/1, 154 (Aminocarbonyl-methyl)-di-tert.-butyl- E2, 22 (l-Amino-ethyl)-hydroxy- E2, 309 (4-Amino-phenyl)-diphcnyl- XII/1, 149 [l-(4-Amino-phenyl)-vinyl]-hydroxy- El, 272 (3-Amino propyloxy) hydroxy El, 319 /<-Anilino benzyl) hvdmxy... 

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