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Homodimers as receptors ligands

FIGURE 18.5 Natural compounds presenting a C2 symmetry axis. [Pg.383]

CHAPTER 18 Homo and Heterodimer Ligands the Twin Drug Approach [Pg.384]

Trans-piperidine derivative DAT / = 228nM SERT /C = 5880nM [Pg.384]

Symmetrical methoctramine polyamine derivatives (nAChR antagonist) [Pg.384]

In the case of enkephalines, dimerization has shown better analgetic properties when compared to their monomeric counterparts (Eigme 18.9). The increase in potency [Pg.385]

See other pages where Homodimers as receptors ligands is mentioned: [Pg.383] [Pg.383]

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A, receptor

Homodimer

Homodimers

Receptor ligands