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Equilibria, dissociation

Table 3. Equilibrium Dissociation Constants for Drug—Receptor Complexes In Vitro... Table 3. Equilibrium Dissociation Constants for Drug—Receptor Complexes In Vitro...
Affinity is the strength of binding of a drag to a receptor. It is quantified by an equilibrium dissociation constant. [Pg.18]

From the equilibrium equations, expressions for the various receptor species can be derived and substituted into Equation 3.32. With conversion of all equilibrium association constants to equilibrium dissociation constants, a general binding expression results for radioactive CD4... [Pg.53]

Converting to equilibrium dissociation constants (i.e., Kd = 1/Ka) leads to the equation... [Pg.75]

It can be seen that the equality defined in Equation 4.32 is true only when ICSo = KB (i.e., the concentration of a non-competitive antagonist that reduces the binding of a tracer ligand by 50% is equal to the equilibrium dissociation constant of the antagonist-receptor complex). [Pg.75]

The equilibrium dissociation constant of the agonist-receptor complex (Ka) can be obtained by a regression of 1/[A] upon 1/[A7]. This leads to a linear regression from which... [Pg.97]


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See also in sourсe #XX -- [ Pg.181 ]

See also in sourсe #XX -- [ Pg.364 , Pg.366 , Pg.417 ]

See also in sourсe #XX -- [ Pg.364 , Pg.366 , Pg.417 ]

See also in sourсe #XX -- [ Pg.24 ]




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Acid dissociation equilibria

Acid-base dissociation equilibria. Strength of acids and bases

Acid-base equilibria percent dissociation

Affinity equilibrium dissociation constant

Agonist dissociation equilibrium constant

Alkali metal halide dimers calculation of equilibrium bond distances and dissociation energies

Appendix 1.2A Equilibrium, Dissociation, and Affinity Constants

Association dissociation equilibrium

Association-Dissociation Equilibria of Enzymes

Association-dissociation equilibrium micellization

Chemical equilibrium ionic dissociation reaction from

Chemical reaction equilibrium dissociation

Constants equilibrium dissociation constant

Counterion dissociation equilibrium

Determination of Bond Dissociation Energies by Thermal Equilibrium Methods

Dissociation and Equilibrium Constants

Dissociation constant The equilibrium

Dissociation equilibria in solution

Dissociation equilibria, glasses

Dissociation equilibrium constant definition

Dissociation equilibrium constant measurement

Dissociation reactions, local equilibrium

Effective dissociation equilibrium constant

Electrolyte dissociation equilibrium

Enzyme association-dissociation equilibria

Equilibrium calculations dissociating species

Equilibrium condition associations/dissociations

Equilibrium constant acid dissociation

Equilibrium constant dissociation

Equilibrium constant electrolyte dissociation

Equilibrium constant for dissociation of weak electrolytes

Equilibrium constant weak electrolyte dissociation

Equilibrium constants base dissociation

Equilibrium dissociation constant dimensions

Equilibrium dissociation energy

Equilibrium for dissociation

Experimental determination of the dissociation equilibrium constant. Ostwalds dilution law

H2CO3, dissociation equilibrium

Influence on Dissociation Equilibria

Intrinsic equilibrium dissociation constant

Kinetic constants dissociation constant Equilibrium

Macroscopic Dissociation Equilibria

Macroscopic equilibrium dissociation constant

Microscopic Dissociation Equilibria

One-Temperature Approach to Vibrational Kinetics and Energy Balance of CO2 Dissociation in Non-Equilibrium Plasma Major Equations

Phosphoric acid dissociation equilibria

Studies equilibrium dissociation

Sulfuric acid dissociation equilibria

Temperature equilibrium dissociation pressure

Thermal equilibrium determination dissociation energies

Water dissociation equilibrium

Weak association and dissociation equilibria of long-chain flotagents

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