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Antagonists allosteric

A. Pi/ erard, Control of the activity of Escherichia coli carbamoyl phosphate synthetase by antagonistic allosteric effectors. Science 154, 1572 1573 (1966). [Pg.241]

Antagonist An antagonist is a receptor ligand preventing the action of an agonist, in a direct (competitive) or indirect (allosteric) manner. [Pg.599]

FIGURE 4.11 Relationship between the observed IC50 for allosteric antagonists and the amount of radioligand present in the assay according to Equation 4.13. Dotted line shows relationship for a competitive antagonist. [Pg.66]

It is assumed that the radioligand [A ] binds to a site separate from one binding an allosteric antagonist [B]. [Pg.75]

Relationship Between IC50 (itid Kifor Allosteric Antagonists... [Pg.76]

The concentration of allosteric antagonist [B] that reduces a signal from a bound amount [A ] of radioligand by 50% is defined as the IC50 ... [Pg.76]

Characterization of the allosteric interactions between antagonists and amiloride at the human ajA-adrenergic receptor. Mol. Pharmacol. 53 916-925. [Pg.78]

See other pages where Antagonists allosteric is mentioned: [Pg.134]    [Pg.65]    [Pg.159]    [Pg.1969]    [Pg.86]    [Pg.152]    [Pg.485]    [Pg.134]    [Pg.65]    [Pg.159]    [Pg.1969]    [Pg.86]    [Pg.152]    [Pg.485]    [Pg.517]    [Pg.551]    [Pg.276]    [Pg.65]    [Pg.65]    [Pg.65]    [Pg.66]    [Pg.66]    [Pg.66]    [Pg.66]    [Pg.67]    [Pg.67]    [Pg.67]    [Pg.74]    [Pg.74]    [Pg.74]    [Pg.75]    [Pg.76]    [Pg.80]    [Pg.99]    [Pg.106]    [Pg.107]    [Pg.108]    [Pg.116]    [Pg.120]    [Pg.127]    [Pg.127]    [Pg.127]    [Pg.128]    [Pg.131]    [Pg.131]    [Pg.132]    [Pg.133]    [Pg.133]    [Pg.133]    [Pg.133]   
See also in sourсe #XX -- [ Pg.62 ]



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