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Adrenergic beta-receptor agonists

Indications Bronchospasm associated with asthma Category Adrenergic beta-receptor agonist Tocolytic Half-life 3-6 hours... [Pg.13]

Indications Diagnostic aid for coronary artery disease Category Adrenergic beta-receptor agonist Half-life 1.8 hours... [Pg.43]

Category Adrenergic beta-receptor agonist Catecholamine ... [Pg.189]

Trade names Aerolone Isopro Isuprel (Hospira) Isuprel Mistometer Isuprel Nebulimetro Saventrine Vapo-lso Indications Bronchospasm, ventricular arrhythmias Category Adrenergic beta-receptor agonist Catecholamine Sympathomimetic Half-life 2.5-5 minutes... [Pg.315]

Just how the calcium alters the effects of adrenaline and dobutamine is not known, but since they are both beta-receptor agonists a reasonable suggestion is that calcium interferes with the signal transduction through the beta-adrenergic receptor complex. The clinical importance of these findings is uncertain. [Pg.890]

CNS inflammation induced by IPS downregulates 1A1 activity in rat loss prevented by beta adrenergic receptor agonist (Abdulla and Renton, 2005). [Pg.57]

Beta agonists. Beta adrenergic receptors can be rapidly down regulated by agonists and if this is desired for an antidepressant action, beta agonists may be useful. To date, it has not been possible to identify beta 1 or beta 2 agonists that successfully penetrate the brain and yet are not cardiotoxic. Pursuing safer beta 1 and beta 2... [Pg.263]

To clarify some of the puzzling differential effects of sympathomimetic drugs on various tissues, in 1948 Ahlquist (76) introduced the concept of two distinct types of adrenergic receptors as defined by their responses to (1), (2), and (17), which he called alpha receptors and beta receptors. Alpha receptors were defined as those that responded in rank order of agonist potency as (2) > (1) (17). Beta receptors were defined as those responding in potency order of (17) > (2) > (1). Subsequently, /3-receptors were further divided into /3i-receptors, located primarily in cardiac tissue, and /32-adrenoceptors, located in smooth muscle and other tissues, given that (1) and (2) are approximately equipotent at cardiac... [Pg.27]

K., Lancaster, M. E., Lee, F, Hart, R., Paulik, M. A., Sherman, B. W, True, T., Cowan, C. Synthesis and evaluation of potent and selective beta(3) adrenergic receptor agonists containing acylsulfonamide, sulfonylsulfonamide, and sulfonylurea carboxylic acid isosteres. J. Med. Chem. 2002,45(3), 567-583. [Pg.336]

M. J., Fisher, M. H., Weber, A. E. 3-Pyridylethanolamines potent and selective human beta 3 adrenergic receptor agonists. Bioorg. Med. Chem. Lett. 1998, S(21), 3087-3092. [Pg.339]

D. Hughes, E. Grabowski, P. Reider, Practical chemoenzymatic synthesis of a pyr-idylethanolamino beta-3 adrenergic receptor antagonist - stereospecific beta-3 agonist used in obesity therapy, produced by yeast-mediated asymmetric reduction of a ketone, Tetrahedron Lett. 1999, 40 (37j, 6739-6743. [Pg.1456]

The side effects of beta-adrenergic receptor agonists are tremor, tachycardia, and palpitations. [Pg.109]

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See also in sourсe #XX -- [ Pg.140 ]



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Adrenergic agonist

Adrenergic receptors receptor

Agonists adrenergic receptors

Beta receptors

Beta-adrenergic-receptor agonists/antagonists

Receptor agonists

Receptor beta adrenergic

Receptors 3-adrenergic

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