Promiscuous inhibitors

McGovern, S. L., Caselli, E., Grigorieff, N., Shoichet, B. K. A common mechanism underlying promiscuous inhibitors from virtual and high-throughput screening. J. Med. Chem. 2002, 45, 1712-1722. 

Grigorieff, N., Shoichet, B.K. A common mechanism underlying promiscuous inhibitors from virtual and high-throughput screening. 

Feng BY, Shelat A, Doman TN, et al. (2005) High-throughput assays of promiscuous inhibitors. Nat. Chem. Biol. 1 146-148. 

Giannetti, A. M., Koch, B. D., and Browner, M. F. (2008). Surface plasmon resonance based assay for the detection and characterization of promiscuous inhibitors. Journal of Medicinal Chemistry 51, 574—580. 

Eliminate reactive functional groups, promiscuous inhibitors, and ... 

Feng, B.Y. and B.K. Shoichet. 2006. A detergent-based assay for the detection of promiscuous inhibitors. Nat. Protoc. 1,550-553. 

Feng BV Shelat A, Doman TN, Guy RK, and Shoichet BK. High-throughput assays for promiscuous inhibitors. Nat Chew, Biol 2005 1 146—148. 

McGovern SL, Caselli E, Grigorieff N, and Shoichet BK. A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening./Med C/tem 2002 45 1712-1722. 

Ryan AJ, Gray NM, Lowe PN, and Chung C-w. Effect of Detergent on Promiscuous Inhibitors./Med Chem2003 46 3448-3451. 

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