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Opioid receptors agonist binding

A 17 amino acid long peptide sequentially related to opioid peptides in particular dynorphin A. OFQ/N is inactive at the 5, k, and p opioid receptors, but binds to its own NOP receptor (formerly ORL-1, for opioid receptor like-1). In contrast to opioid peptides, OFQ/N has no direct analgesic properties. OFQ/N is the first example for the discovery of a novel neurotransmitter from tissue extracts by using an orphan receptor as bait. Centrally administered in rodents, OFQ/N exerts anxiolytic properties. OFQ/N agonists and antagonists... [Pg.917]

Randic, M., Cheng, G., and Kojic, L. (1995). Kappa-opioid receptor agonists modulate excitatory transmission in substantia gelatinosa neurons of the rat spinal cord. J. Neurosci. 15, 6809-6826. Ransom, R. W., and Stec, N. L. (1988). Cooperative modulation of [3H] MK-801 binding to the jV-methyl-D-aspartate receptor-ion channel complex by L-glutamate, glycine, and polyamines. [Pg.202]

Spetea M, Toth F, Schiitz J, Otvos F, Toth G, Benyhe S, Borsodi A, Schmidhammer H (2003) Binding characteristics of [3H] 14-methoxymetopon, a high affinity p-opioid receptor agonist. Eur J Neurosci 18 290-295... [Pg.89]

Kane BE, Nieto MJ, McCurdy CR, Ferguson DM (2006) A unique binding epitope for salvinorin A, a non-nitrogenous kappa opioid receptor agonist. FEBS J 273 1966-1974... [Pg.305]

Mfller, D.K., J.R. Lever, K.R. Rodvelt, et al. 2007. LobeUne, a potential pharmacotherapy for drug addiction, binds to mu opioid receptors and diminishes the effects of opioid receptor agonists. Drug Alcohol Depend. 89(2-3) 282-291. [Pg.531]

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See also in sourсe #XX -- [ Pg.90 ]



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Agonist binding

Opioid agonists

Opioid receptor binding

Opioid receptors

Opioids agonists

Opioids receptor agonists

Opioids receptors

Receptor agonist binding

Receptor agonists

Receptor binding

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