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Muscarinic receptor agonists gastrointestinal effects

CI-979 (29) is a balanced muscarinic agonist having equal affinities for cloned ml and m2 receptors (144). However, unlike prototypical muscarinic compounds such as (25), (29) increases central muscarinic tone, as indicated by behavioral and electroencephalogram (EEG) parameters, at doses lower than those requited to produce gastrointestinal effects (144). CI-979 is well tolerated in humans up to a dose of 1 mg. Dose-limiting side effects such as stomach pain and emesis were observed at a dose of 2 mg. [Pg.99]


See other pages where Muscarinic receptor agonists gastrointestinal effects is mentioned: [Pg.106]    [Pg.180]    [Pg.227]    [Pg.120]    [Pg.470]    [Pg.150]    [Pg.775]    [Pg.212]    [Pg.299]   
See also in sourсe #XX -- [ Pg.115 , Pg.116 ]




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Agonist effect

Muscarin

Muscarine

Muscarine receptors

Muscarines

Muscarinic

Muscarinic agonists

Muscarinic receptor agonists

Muscarinic receptors

Muscarinics

Receptor agonists

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