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Metabolism in drug discovery

Kumar GN, Surapaneni S (2001) Role of drug metabolism in drug discovery and development. Med Res Rev 21 397—411... [Pg.499]

Lin JH, Lu AYH. Role of pharmacokinetics and metabolism in drug discovery and metabolism. Pharmacol Rev 1997 49 403-49. [Pg.94]

Komura H, Kawahara I, Shigemoto Y, et al. High throughput screening of pharmacokinetics and metabolism in drug discovery (I)—establishment of assessment system for absorption to compounds with a wide diversity of physical properties. Yakugiu Zasshi 2005 Jan 125(1) 121-130. [Pg.163]

Gibbs, J. P., Hyland, R., and Youdim, K. (2006) Minimizing polymorphic metabolism in drug discovery evaluation of the utility of in vitro methods for predicting pharmacokinetic consequences associated with CYP2D6 metabolism. Drug Metab. Dispos. 34, 1516-1522. [Pg.38]

Pharmacokinetics and Metabolism in Drug Discovery and Preclinical Development... [Pg.57]

Mitigating heterocycle metabolism in drug discovery 12JMC6002. Modification of biologically active plant metabolites via the metal complex catalysis reactions as a promising direction in medicinal chemistry 13IZV605. [Pg.256]

Jean DJ St Jr, Fotsch C (2012) Mitigating heterocycle metabolism in drug discovery. J Med Chem 55(13) 6002-6020... [Pg.320]

Patten, C. J. New technologies for assessing UDP-glucuronosyltransferase (UGT) metabolism in drug discovery and development. Drug Discovery Today 2006, 3, 73-78. [Pg.822]


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See also in sourсe #XX -- [ Pg.2263 ]




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