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Is a Paradigm Shift in Drug Discovery Imminent

Dancey J, Sausville EA (2003) Issues and progress with protein kinase inhibitors for cancer treatment. Nat Rev Drug Discov 2 296-313 [Pg.184]

Levitski A, Gazit A (1995) Tyrosine kinase inhibition An approach to drug development. Science 267 1782-1788 [Pg.184]

Tibes R, Trent J, Kurzrock R (2005) Tyrosine kinase inhibitors and the dawn of molecular cancer therapeutics. Annu Rev Pharmacol Toxicol 45 357-384 [Pg.184]

Gibbs J, Oliff A (1994) Pharmaceutical research in molecular oncology. Cell 79 193-198 [Pg.184]

Donato NJ, Talpaz M (2000) Clinical use of tyrosine kinase inhibitors Therapy for chronic myelogenous leukemia and other cancers. Clin Cancer Res 6 2965-2966 [Pg.184]


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