Big Chemical Encyclopedia

Chemical substances, components, reactions, process design ...

Articles Figures Tables About

Strong agonist

Morphine p agonist— strong (full) +++ +++ +++ Prototype of the class, marked sedation, poor oral bioavailability, histamine release... [Pg.159]

Methadone p agonist— strong (full) + ++ +++ +++ Oral activity and j long duration, useful in r. maintenance... [Pg.159]

Meperidine p agonist-strong (full) +++ +++ +++ M blocker (no miosis or smooth muscle contraction), forms normeperidine h> possible seizures... [Pg.159]

Synthetic steroid with strong glucocorticoid-agonistic activity. Dexamethasone is over 10 times more potent than cortisol due to a higher binding affinity for glucocorticoid receptor and a decreased clearance rate of the compound. Due to its potency, dexamethasone is widely used in the clinics for the treatment of inflammatory diseases. [Pg.422]

In another example from the literature [40], we see a strong correlation between potency and PSA. In this case a series of 53 CCR5 receptor agonists have been... [Pg.446]

See other pages where Strong agonist is mentioned: [Pg.57]    [Pg.350]    [Pg.130]    [Pg.228]    [Pg.57]    [Pg.350]    [Pg.130]    [Pg.228]    [Pg.242]    [Pg.258]    [Pg.382]    [Pg.384]    [Pg.219]    [Pg.156]    [Pg.22]    [Pg.41]    [Pg.453]    [Pg.713]    [Pg.835]    [Pg.891]    [Pg.907]    [Pg.1047]    [Pg.1276]    [Pg.8]    [Pg.81]    [Pg.93]    [Pg.147]    [Pg.230]    [Pg.172]    [Pg.150]    [Pg.184]    [Pg.207]    [Pg.246]    [Pg.387]    [Pg.16]    [Pg.44]    [Pg.105]    [Pg.158]    [Pg.199]    [Pg.266]    [Pg.369]    [Pg.328]    [Pg.402]    [Pg.304]    [Pg.344]    [Pg.23]    [Pg.373]   
See also in sourсe #XX -- [ Pg.135 , Pg.136 , Pg.137 , Pg.138 , Pg.139 ]



SEARCH



© 2024 chempedia.info