Reactivation potency, acetylcholinesterase

Jun, D., Musilova, L., Lazenska, H., Kuca, K., Kassa, J., Bajgar, J. (2007). Potency of several oximes to reactivate human acetylcholinesterase and hutyrylcholinesterase inWhited by paraoxon and methyl-paraoxon in vitro. The IXth International Meeting on Cholinesterases. Suzhou, CWna, May 6-10, 2007. Program Book, p. 140. 

Kuca, K., Cabal, J., Jun, D., Kassa, K., Bartosova, L., Kunesova, G. (2005c). In vitro reactivation potency of some acetylcholinesterase reactivators against sarin and cyclosarin-induced inhibitions. J. Appl. Toxicol. 25 296-300. 

Yang, G.Y., Oh, K.A., Park, N.J., Jung, Y.S. (2007). New oxime reactivators connected with CH20(CH2) 0CH2 linker and their reactivation potency for organophosphorus agents-inhibited acetylcholinesterase. Bioorg. Med. Chem. 15 7704-10. 

W14. Worek, F., Widmann, R., Knopff, O., and Szinicz, L., Reactivating potency of obidoxime, pralidoxime, HI 6 and Hlo 7 in human erythrocyte acetylcholinesterase inhibited by highly toxic organophosphorus compounds. Arch. Toxicol. 72, 237-243 (1998). 

Milatovic, D., and Vorkapic-Furac, J., 1989. Synthesis of three pyridoxal oxime derivatives and their reactivating potency against phosphylated acetylcholinesterase. Acta Pharmaceutica Jugoslavia. 39 281-287. 

Jeong, H.C., Kang, N.S., Park, N.J., et ak, 2009. Reactivation potency of fluori-nated pyridinium oximes for acetylcholinesterases inhibited by paraoxon organophosphorus agent. Bioorg. Med. Chem. Lett. 19, 1214-1217. 

Oh, K. A., Park, N.J., Park, N.S., et al., 2008. Determination of reactivation potency for DFP- and paraoxon-inhibited acetylcholinesterases by pyridinium oximes. Chem. Biol. Interact. 175, 365-367. 

Kuca, K., Cabal, J., Jim, D., Hrahinova, M. (2007). Potency of five structurally different acetylcholinesterase reactivators to reactivate human brain cholinesterases inhibited by cyclosarin. Clin. Toxicol. (Phila.) 45 512-15. 

Kuca, K., Picha, J., Cabal, J., Liska, F. (2004b). Synthesis of the three monopyridinium oximes and evaluation of their potency to reactivate acetylcholinesterase inhibited by nerve agents. J. Appl. Biomed. 2 51-6. 

Musilek, K., Lipka, L., Racakova, V., Kuca, K., Jun, D., Dohnal, V., Dolezal, V. (2006b). New methods in synthesis of acetylcholinesterase reactivators and evaluation of their potency to reactivate cyclosarin-inhibited AChE. Chem. Papers 60 48-51. 

Odzak, R., Calic, M., Hrenar, T., Primozic, I., Kovarik, Z. (2007). Evaluation of monoquatemary pyridinium oximes potency to reactivate tabun-inhibited human acetylcholinesterase. Toxicology 233 85-96. 

Kuda, K., Cabal, J., Kassa, J., et al, 2005. A comparison of the potency of the oxime HL5-7 and currently used oximes (HI-6, pralidoxime, obidoxime) to reactivate nerve agent-inhibited rat brain acetylcholinesterase by in vitro methods. Acta Medica (Hradec Kralove) 48, 81-86. 

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