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Preparation of Immunotoxin Conjugates via Amine- and Sulfhydryl-Reactive Heterobifunctional Cross-linkers

Preparation of Immunotoxin Conjugates via Amine- and Sulfhydryl-Reactive Heterobifunctional Cross-linkers [Pg.516]

To make effective immunotoxin conjugates using the following cross-linkers, it is necessary to cross-link intact A—B toxins to antibodies, not single-chain or A-chain toxins. Using intact two-subunit toxins allows the A chain to break free of the complex [Pg.516]




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Aminals, preparation

Amination, 15 preparation

Amine conjugating

Amines preparation

Amines reactivities

Conjugate preparation

Conjugated reactivity

Conjugation amine

Conjugation cross

Cross preparation

Cross reactivity

Cross-conjugated

Cross-linker

Heterobifunctional

Heterobifunctional cross-linkers

Immunotoxin

Immunotoxin conjugate

Immunotoxin conjugates preparation

Immunotoxin cross-linkers

Immunotoxin preparation

Immunotoxins

Linker amine

Preparation of Immunotoxin Conjugates

Preparation of conjugates

Preparation of linker

Reactive amines

Sulfhydryls

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