AMPA receptors structure

Kuner, T., Beck, C., Sakmann, B., and Seeburg, R H., Channel-lining residues of the AMPA receptor M2 segment structural environment of the Q7R site and identification of the selective filter, J. Neurosci., 21, 4162 1172, 2001. 

Higuchi, M., Single, F. N., Kohler, M. et al. RNA editing of AMPA receptor subunit GluRB a base-paired intron-exon structure determines position and efficiency. Cell 75 1361-1370,1993. 

Hogner, A., Kastrup, J. S Jin, R., Liljefors, T Mayer, M. L., Egebjerg, J., et al. (2002) Structural basis for AMPA receptor activation and ligand selectivity crystal structures of five agonist complexes with the GluR2 binding core../. Mol. Biol. 322,93-109. 

Fig. 2.5 Structures of kainate and AMPA receptor antagonists. LY382884 (a) and LY382884 diethyl ester (b) are kainate receptor antagonists CP-465022 (c), GYKI 52466 (d) CFM-2 (e) and GYKI 53655 (R= CONHMe) (f) are AMPA receptor antagonists...

Structure and Distribution of AMPA Receptor Subunits in Brain... 

Ornstein, P. L., Arnold, M. B., Augenstein, N. K., Lodge, D., Leander, J. D., Schoepp, D. D. (3SR,4aRS,6RS,8aRS)-6-[2-(li7-tetrazol-5-yl)ethyl]decahydroisoquinoline-3-carboxylic acid a structurally novel, systematically active, competitive AMPA receptor antagonist. J. Med. Chem. 1993, 36, 2046-2048. 

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